| Name | A 366 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 2753 |
| Prices | $189.00, $765.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Cas Number | 1527503-11-2 |
| Chemical Name | 5'-Methoxy-6'-[3-(1-pyrrolidinyl)propoxy]spiro[cyclobutane-1,3'-[3H]indol]-2'-amine |
| Formula | C19H27N3O2 |
| Molecular Weight | 329.44 |
| Purity | >98 % |
| Description | Potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC 50 = 3.3 nM). Exhibits >1000-fold selectivity for G9a/GLP over 21 other methyltransferases. Decreases levels of lysine 9 dimethylation on histone H3 (H3K9Me2) in PC3 cells. |
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