AGN 193109

Name AGN 193109
Supplier Tocris Bioscience
Catalog 1072
Prices $269.00
Sizes 10 mg
Function Type Antagonist
Cas Number 171746-21-7
Chemical Name 4-[2-[5,6-Dihydro-5,5-dimethyl-8-(4-methylphenyl)-2-naphthalenyl]ethynyl]benzoicacid
Formula C28H24O2
Molecular Weight 392.49
Purity >97 %
Description High affinity pan-retinoic acid receptor (RAR) antagonist (K d values are 2, 2 and 3 nM at RAR α , RAR β and RAR γ , respectively). Does not bind retinoic X receptors.
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Product References

Structure activity relationships of a series of buspirone analogs at alpha-1 - Structure activity relationships of a series of buspirone analogs at alpha-1

Saussy DL Jr, Goetz AS, Queen KL, King HK, Lutz MW, Rimele TJ. J Pharmacol Exp Ther. 1996 Jul;278(1):136-44.

Failure of AH11110A to functionally discriminate between alpha(1)-adrenoceptor - Failure of AH11110A to functionally discriminate between alpha(1)-adrenoceptor

Eltze M, Konig H, Ullrich B, Grebe T. Eur J Pharmacol. 2001 Mar;415(2-3):265-76.