[Pyr 1 ]-Apelin-13

Name [Pyr 1 ]-Apelin-13
Supplier Tocris Bioscience
Catalog 1208
Prices $175.00
Sizes 1 mg
Cas Number 217082-60-5
Formula C69H108N22O16S
Molecular Weight 1533.81
Description Highly potent pyroglutamyl form of apelin-13. Endogenous ligand for apelin APJ receptor (EC 50 = 0.37 nM) that displays potent vascular effects in vivo .
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Product References

[(125)I]-(Pyr(1))Apelin-13 is a novel radioligand for localizing the APJ orphan - [(125)I]-(Pyr(1))Apelin-13 is a novel radioligand for localizing the APJ orphan

Katugampola SD, Maguire JJ, Matthewson SR, Davenport AP. Br J Pharmacol. 2001 Mar;132(6):1255-60.

Central and peripheral cardiovascular actions of apelin in conscious rats. - Central and peripheral cardiovascular actions of apelin in conscious rats.

Kagiyama S, Fukuhara M, Matsumura K, Lin Y, Fujii K, Iida M. Regul Pept. 2005 Feb 15;125(1-3):55-9.

Emerging roles of apelin in biology and medicine. - Emerging roles of apelin in biology and medicine.

Kleinz MJ, Davenport AP. Pharmacol Ther. 2005 Aug;107(2):198-211.