| Name | ARC 239 dihydrochloride |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 4890 |
| Prices | $139.00, $585.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Antagonist |
| Cas Number | 55974-42-0 |
| Chemical Name | 2-[2-(4-(2-Methoxyphenyl)piperazin-1-yl)ethyl]-4,4-dimethyl-1,3-(2H,4H)-isoquinolindionedihydrochloride |
| Formula | C24H29N3O3.2HCl |
| Molecular Weight | 480.43 |
| Purity | >98 % |
| Description | Selective α 2B adrenoceptor antagonist (pK D values are 8.8, 6.7 and 6.4 at α 2B , α 2A , and α 2D receptors respectively). Also available as part of the α 2 -Adrenoceptor Tocriset™ . |
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Fuder H, Selbach M. Naunyn Schmiedebergs Arch Pharmacol. 1993 Apr;347(4):394-401.