Name | ASP 2535 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 3737 |
Prices | $235.00 |
Sizes | 10 mg |
Function Type | Inhibitor |
Cas Number | 374886-51-8 |
Chemical Name | 4-[3-(1-Methylethyl)-5-(6-phenyl-3-pyridinyl)-4H-1,2,4-triazol-4-yl]-2,1,3-benzoxadiazole |
Formula | C22H18N6O |
Molecular Weight | 382.42 |
Purity | >98 % |
Description | Potent and selective GlyT1 inhibitor (IC 50 = 92 nM). Exhibits 50-fold selectivity over GlyT2. Attenuates MK 801 -induced working memory deficits and PCP -induced visual learning deficits in mice. Orally available and brain penetrant. |
Supplier Page | Shop |