| Name | ATC 0065 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 3531 |
| Prices | $205.00 |
| Sizes | 10 mg |
| Function Type | Antagonist |
| Cas Number | 510732-84-0 |
| Chemical Name | N2-[cis-4-[[2-[4-Bromo-2-(trifluoromethoxy)phenyl]ethyl]amino]cyclohexyl]-N4,N4-dimethyl-2,4-quinazolinediaminedihydrochloride |
| Formula | C25H29BrF3N5O.2HCl |
| Molecular Weight | 625.35 |
| Purity | >98 % |
| Description | Orally active, potent and selective melanin-concentrating hormone receptor 1 (MCH 1 ) antagonist (IC 50 = 15.7 nM) that displays > 96-fold selectivity over MCH 2 . Exhibits antidepressant and anxiolytic activity in vivo . Also displays affinity for 5-HT 1A and 5-HT 2B receptors (IC 50 values are 62.9 and 266 nM respectively). |
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