Name | AZ 191 |
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Supplier | Tocris Bioscience |
Catalog | 4832 |
Prices | $179.00, $745.00 |
Sizes | 10 mg, 50 mg |
Function Type | Inhibitor |
Cas Number | 1594092-37-1 |
Chemical Name | N-[2-Methoxy-4-(4-methyl-1-piperazinyl)phenyl]-4-(1-methyl-1H-pyrrolo[2,3-c]pyridin-3-yl)-2-pyrimidinamine |
Formula | C24H27N7O |
Molecular Weight | 429.52 |
Purity | >98 % |
Description | Potent DYRK1B inhibitor (IC 50 values are 17, 88 and 1890 nM for DYRK1B, DYRK1A and DYRK2 respectively). Inhibits DYRK1B-induced G i phase cell cycle arrest in Panc-1 cells in vitro . |
Supplier Page | Shop |