CGP 52432

• Supplier: Tocris Bioscience
• Catalog: 3360
• Prices: $199.00, $825.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 139667-74-6
• Chemical Name: 3-[[(3,4-Dichlorophenyl)methyl]amino]propyl]diethoxymethyl)phosphinicacid
• Formula: C15H24Cl2NO4P
• Molecular Weight: 384.24
• Purity: >99 %
• Description: Potent, selective GABA B receptor antagonist (IC 50 = 85 nM).

Product References

CGP 52432: a novel potent and selective GABAB autoreceptor antagonist in rat - CGP 52432: a novel potent and selective GABAB autoreceptor antagonist in rat

Lanza M, Fassio A, Gemignani A, Bonanno G, Raiteri M. Eur J Pharmacol. 1993 Jun 24;237(2-3):191-5.

GABA(B) receptors as potential targets for drugs able to prevent excessive - GABA(B) receptors as potential targets for drugs able to prevent excessive

Bonanno G, Fassio A, Sala R, Schmid G, Raiteri M. Eur J Pharmacol. 1998 Dec 4;362(2-3):143-8.

Blockade of GABA(B) receptors facilitates muscarinic agonist-induced epileptiform - Blockade of GABA(B) receptors facilitates muscarinic agonist-induced epileptiform

Libri V, Constanti A, Postlethwaite M, Bowery NG. Naunyn Schmiedebergs Arch Pharmacol. 1998 Aug;358(2):168-74.