CI 966 hydrochloride

• Supplier: Tocris Bioscience
• Catalog: 2942
• Prices: $189.00, $765.00
• Sizes: 10 mg, 50 mg
• Function Type: Inhibitor
• Cas Number: 110283-66-4
• Chemical Name: 1-[2-[bis[4-(Trifluoromethyl)phenyl]methoxy]ethyl]-1,2,5,6-tetrahydropyridine-3-carboxylicacidhydrochloride
• Formula: C23H21F6NO3.HCl
• Molecular Weight: 509.87
• Purity: >98 %
• Description: Selective inhibitor of the GABA transporter GAT-1 (IC 50 values are 0.26 and 1.2 μ M at cloned human and rat GAT-1 respectively). Displays over 200-fold selectivity over GAT-2 and GAT-3. Centrally active upon systemic administration in vivo . Anticonvulsive and neuroprotective.

Product References

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