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α -Conotoxin ImI

Name α -Conotoxin ImI
Supplier Tocris Bioscience
Catalog 1085
Prices $239.00
Sizes 500 µg
Function Type Antagonist
Cas Number 156467-85-5
Formula C52H78N20O15S4
Molecular Weight 1351.6
Description Nicotinic receptor antagonist that displays selectivity for homomeric α 7 and α 9 receptors (IC 50 values are 220 and 1800 nM respectively). Displays no effect on α 2 β 2, α 3 β 2, α 4 β 2, α 2 β 4, α 3 β 3 and α 4 β 4 subunit combinations.
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Product References

A nicotinic acetylcholine receptor ligand of unique specificity, alpha-conotoxin - A nicotinic acetylcholine receptor ligand of unique specificity, alpha-conotoxin

McIntosh JM, Yoshikami D, Mahe E, Nielsen DB, Rivier JE, Gray WR, Olivera BM. J Biol Chem. 1994 Jun 17;269(24):16733-9.

alpha-Conotoxin ImI exhibits subtype-specific nicotinic acetylcholine receptor - alpha-Conotoxin ImI exhibits subtype-specific nicotinic acetylcholine receptor

Johnson DS, Martinez J, Elgoyhen AB, Heinemann SF, McIntosh JM. Mol Pharmacol. 1995 Aug;48(2):194-9.

Alpha-conotoxin-ImI: a competitive antagonist at alpha-bungarotoxin-sensitive - Alpha-conotoxin-ImI: a competitive antagonist at alpha-bungarotoxin-sensitive

Pereira EF, Alkondon M, McIntosh JM, Albuquerque EX. J Pharmacol Exp Ther. 1996 Sep;278(3):1472-83.



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