(±)-CP 47497

• Supplier: Tocris Bioscience
• Catalog: 3780
• Prices: $139.00, $585.00
• Sizes: 10 mg, 50 mg
• Function Type: Agonist
• Cas Number: 70434-82-1
• Chemical Name: rel-5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3-hydroxycyclohexyl]phenol
• Formula: C21H34O2
• Molecular Weight: 318.49
• Purity: >98 %
• Description: Potent CB 1 receptor agonist (K i = 2.2 nM). Exhibits analgesic, motor depressant, anticonvulsant and hypothermic effects in vivo .

Product References

Cannabimimetic activity from CP-47,497, a derivative of 3-phenylcyclohexanol. - Cannabimimetic activity from CP-47,497, a derivative of 3-phenylcyclohexanol.

Weissman A, Milne GM, Melvin LS Jr. J Pharmacol Exp Ther. 1982 Nov;223(2):516-23.

Structure-activity relationships for cannabinoid receptor-binding and analgesic - Structure-activity relationships for cannabinoid receptor-binding and analgesic

Melvin LS, Milne GM, Johnson MR, Subramaniam B, Wilken GH, Howlett AC. Mol Pharmacol. 1993 Nov;44(5):1008-15.

Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940. - Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940.

Huffman JW, Thompson AL, Wiley JL, Martin BR. Bioorg Med Chem. 2008 Jan 1;16(1):322-35. Epub 2007 Sep 22.